Found 92 recordings
DICL IDIon ChannelCompound FunctionSpeciesValueReferences
DICL_CP_0316539Gamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2Allosteric ModulatorRattus norvegicus (Rat)Ki: >15000 nM10.1016/j.bmcl.2020.127536, 32898695
DICL_CP_0319565Gamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2Allosteric ModulatorRattus norvegicus (Rat)Ki: 972 nM10.1016/j.bmcl.2020.127536, 32898695
DICL_CP_0319792Gamma-aminobutyric acid receptor subunit alpha-5/beta-1-3/gamma-2LInactiveRattus norvegicus (Rat)Inhibition: No effect10.1111/j.1476-5381.2011.01604.x, 21797842
DICL_CP_0323088Gamma-aminobutyric acid receptor subunit alpha-5/beta-1-3/gamma-2LInactiveRattus norvegicus (Rat)Inhibition: No effect10.1016/j.bcp.2011.09.002, 21924247
DICL_CP_0323752Gamma-aminobutyric acid receptor subunit alpha-5/beta-2/gamma-2Inverse AgonistRattus norvegicus (Rat)Ki: 9 nM10.1016/j.bmc.2007.01.053, 17306981
DICL_CP_0326172Gamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2 ModulatorRattus norvegicus (Rat)Ki: 740 nM10.1021/jm020999w, 12519068
DICL_CP_0326174Gamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2 ModulatorRattus norvegicus (Rat)Ki: 210 nM10.1021/jm020999w, 12519068
DICL_CP_0326214Gamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2Allosteric ModulatorRattus norvegicus (Rat)Ki: 459 nM10.1016/j.bmcl.2020.127536, 32898695
DICL_CP_0327635Gamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2 ModulatorRattus norvegicus (Rat)Ki: 223 nM10.1021/jm020999w, 12519068
DICL_CP_0327737Gamma-aminobutyric acid receptor subunit alpha-5/beta-3/gamma-2AgonistRattus norvegicus (Rat)Ki: 520 nM10.1021/jm031076j, 15084116
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